Derivatives
Mostrando 13-24 de 6480 artigos, teses e dissertações.
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13. Novel Insecticides from Alkylated and Acylated Derivatives of Thymol and Eugenol for the Control of Plutella xylostella (Lepidoptera: Plutellidae)
Plutella xylostella cause considerable harm to the production of broccoli, Chinese cabbage, cabbage and cauliflower. The control of P. xylostella is mainly performed using commercial insecticides, which have even led to the emergence of resistant populations. Two easily available natural products found in different plants essential oil, thymol and eugenol, s
Journal of the Brazilian Chemical Society. Publicado em: 2022
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14. Synthesis and Anti-Chikungunya Virus (CHIKV) Activity of Novel 1,4-Naphthoquinone Sulfonamide and Sulfonate Ester Derivatives
Chikungunya virus (CHIKV) is a re-emerging disease caused by an alphavirus of the Togaviridae family. Since its first description in 1952, the disease has spread worldwide, affecting populations in both tropical and temperate countries. To date, there is no licensed vaccine or specific pharmacological treatment. Therefore, there is an increasing urgency in d
Journal of the Brazilian Chemical Society. Publicado em: 2022
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15. Natural and Semisynthetic Triterpenes from Combretum leprosum Mart. with Antiplasmodial Activity
Malaria is responsible for thousands of deaths each year. Currently, artemisinin combination therapy (ACT) is used as first-choice medication against the disease. However, the emergence of resistant strains prompts the search for alternative compounds. The present study aimed to investigate the antiplasmodial activities of natural triterpenes (compounds 1 an
Journal of the Brazilian Chemical Society. Publicado em: 2022
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16. Benzophenone Derivatives Showed Dual Anti-Inflammatory and Antiproliferative Activities by Inhibiting COX Enzymes and Promote Cyclin E Downregulation
Considering the promising antitumor effects of compounds with dual anti-inflammatory and antiproliferative activities, thus benzophenones analogs (2-7) were evaluated on in vivo anti-inflammatory assay and molecular docking analysis. Those with the best molecular docking results were in vitro evaluated on cyclooxygenase (COX) enzymes and tested regarding ant
Journal of the Brazilian Chemical Society. Publicado em: 2022
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17. ARTEMISININA E DERIVADOS: DESCOBERTA, ESTRATÉGIAS SINTÉTICAS E OBTENÇÃO INDUSTRIAL
Artemisinin, a natural sesquiterpene isolated from the Artemisia annua L. plant, represents a remarkable achievement in the treatment against malaria. Since its discovery in the 1970’s, researchers readily started synthesizing this complex natural product containing an unusual endoperoxide fragment. Despite various total syntheses reported, only in the las
Química Nova. Publicado em: 2022
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18. A New Synthetic Route and Comprehensive Topological Study of a Benzimidazole Derivative
Benzimidazole and its derivatives are molecules that have diverse biological properties, therefore we synthesized and studied a new benzimidazole to understand their physical/chemical properties. The compound was obtained through a new synthetic route, using graphite oxide, in the absence of solvent, with crystalline packaging supported by C-H…N and C-H…
Journal of the Brazilian Chemical Society. Publicado em: 2022
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19. Heteroannulation Reaction of α-Aminoketones for the Efficient Synthesis of 4-Imidazolin-2-ones and 2-Thiones
The hydrogenation of α-oximinoketones in methanol/HCl afforded α-aminoketones, which were applied without purification to the synthesis of 4-imidazolin-2-ones and 2-thiones, including chiral derivatives. The latter two series were obtained in high yields by a heteroannulation reaction of α-aminoketones with isocyanates and isothiocyanates, respectively. A
Journal of the Brazilian Chemical Society. Publicado em: 2022
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20. Volatile Constituents of Floral Scents from Encyclia cordigera (Kunth) Dressler and E. randii (Barb. Rodr.) Porto & Brade (Orchidaceae)
Encyclia cordigera is native from Central America tropical region, and Encyclia randii occurs at Brazilian Amazon environment domains. Floral concentrates from both Encyclia species were extracted, analyzed by gas chromatography-mass spectrometry, and identified compounds belong to terpenoids, phenylpropanoids, and fatty acid derivatives classes. Primary con
Journal of the Brazilian Chemical Society. Publicado em: 2022
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21. Comparative Study of Some Numerical Schemes for a Fractional Order Model of HIV Infection Treatment
ABSTRACT A fractional order mathematical model that already exists in the literature, was considered. This model was established to study the effects of medicinal treatment in people infected with the human immunodeficiency virus (HIV). The importance of this study is that the model evaluates, among other parameters, the density of healthy and HIV-infected C
Trends in Computational and Applied Mathematics. Publicado em: 2022
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22. Using nonlinear models to define production, production rate, and precocity of strawberry cultivars
ABSTRACT The aim of this study was to evaluate, using logistic model, the differences in early production, production rate and total productivity of two strawberry cultivars with transplants from different origins grown in substrate. The experiment was carried out in a randomized block design (RBD), with two strawberry cultivars (Albion and Camarosa) and two
Revista Ceres. Publicado em: 2022
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23. Effects of chemical straighteners on the hair shaft and scalp
Abstract Background The effects of chemical straighteners on the scalp and hair shaft are not fully known, although such substances are widely used. Hair straightening became popular in Brazil with the use of formaldehyde and its derivatives, despite the prohibition by the current legislation. Objective To identify changes in hair shaft and scalp caused by
Anais Brasileiros de Dermatologia. Publicado em: 2022
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24. CLOROFILA EXTRAÍDA DE RESÍDUO INDUSTRIAL DA ERVA-MATE (Ilex paraguaiensis) UMA POSSIBILIDADE DE ECONOMIA CIRCULAR
Chlorophyll is the most abundant green pigment on the planet, it is unstable and decomposes naturally. Mate-herb is a traditional native plant in the southern region of South America, and its tea is part of the local culture and extractive agriculture. The mate-herb industry generates as a by-product a resinous material rich in chlorophyll whose use is propo
Química Nova. Publicado em: 2022